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FK866
CAS No. 658084-64-1
FK866 ( APO866, Daporinad )
Catalog No. M15502 CAS No. 658084-64-1
FK866 (APO866, Daporinad) effectively inhibits nicotinamide phosphoribosyltransferase (NMPRTase) with IC50 of 0.09 nM in a cell-free assay. Phase 1/2.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 32 | In Stock |
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| 5MG | 53 | In Stock |
|
| 10MG | 87 | In Stock |
|
| 25MG | 178 | In Stock |
|
| 50MG | 348 | In Stock |
|
| 100MG | 528 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameFK866
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NoteResearch use only, not for human use.
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Brief DescriptionFK866 (APO866, Daporinad) effectively inhibits nicotinamide phosphoribosyltransferase (NMPRTase) with IC50 of 0.09 nM in a cell-free assay. Phase 1/2.
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DescriptionFK866 (APO866, Daporinad) effectively inhibits nicotinamide phosphoribosyltransferase (NMPRTase) with IC50 of 0.09 nM in a cell-free assay. Phase 1/2.
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SynonymsAPO866, Daporinad
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PathwayMetabolic Enzyme/Protease
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TargetTransferase
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RecptorNMPRTase
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Research AreaCancer
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IndicationSkin Cancer
Chemical Information
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CAS Number658084-64-1
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Formula Weight391.51
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Molecular FormulaC24H29N3O2
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Purity>98%(HPLC)
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SolubilityEthanol: 78 mg/mL (199.22 mM)
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SMILESC1CN(CCC1CCCCNC(=O)/C=C/C2=CN=CC=C2)C(=O)C3=CC=CC=C3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Nahimana A, et al. Blood, 2009, 113(14), 3276-3286.
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